阿培利司盐酸盐
Alpelisib hydrochloride
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基本信息
中文名称阿培利司盐酸盐
英文名称 Alpelisib hydrochloride
CAS号1584128-91-5
分子式C19H23ClF3N5O2S
分子量477.93
储存条件Store in a dry and dark sealed container, short-term (weeks to months) storage at 0-4 ℃, long-term (months to years) storage at -20 ℃.
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Alpelisib hydrochloride (BYL-719 hydrochloride) is a potent, orally active, and selective PI3Kα inhibitor with IC50s of 5 nM, 250 nM, 290 nM and 1200 nM for p110α, p110γ, p110δ, and p110β, respectively. Alpelisib hydrochloride (BYL-719 hydrochloride) shows antineoplastic activity.


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阿培利司盐酸盐