CEP-28122 mesylate salt
CEP-28122 mesylate salt (Synonyms:CEP-28122 (Mesylate salt))
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中文名称CEP-28122 mesylate salt
英文名称 CEP-28122 mesylate salt (Synonyms:CEP-28122 (Mesylate salt))
CAS号2070009-30-0
分子式C29H39ClN6O6S
分子量635.17
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CEP-28122 mesylate salt, a diaminopyrimidine derivative, is a potent, selective, and orally bioavailable ALK inhibitor, with an IC50 value of 1.9 nM for recombinant ALK kinase activity. CEP-28122 has antitumor activity in experimental models of ALK-positive human cancers. CEP-28122 mesylate salt has good pharmacodynamic and pharmacokinetic activity.

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