辛波莫德半富马酸盐
Siponimod Hemifumarate (Synonyms: BAF-312 Hemifumarate)
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3-5days
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¥1166.00
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¥1800.00
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基本信息
中文名称辛波莫德半富马酸盐
英文名称 Siponimod Hemifumarate (Synonyms: BAF-312 Hemifumarate)
CAS号1234627-85-0
分子式C29H35F3N2O3·1/2C4H4O4
分子量574.63 | 516.61(free)
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Siponimod (BAF-312) hemifumarate is a potent and selective sphingosine-1-phosphate (S1P) receptor modulator. Siponimod hemifumarate is selective for S1P1 and S1P5 receptors over S1P2, S1P3, and S1P4 (EC50s of 0.39, 0.98, >10000, >1000, and 750 nM, respectively). Siponimod hemifumarate can be used for multiple sclerosis (MS) research.
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相关文献
PMID: 30621015 PMCID: PMC6356776 DOI: 10.3390/cells8010024
PMID: 30038666 PMCID: PMC6050809 DOI: 10.1177/1756286418788013
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