富马酸沃诺拉赞 | 富马酸伏诺拉生| 1260141-27-2
Vonoprazan Fumarate | TAK-438
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基本信息
中文名称富马酸沃诺拉赞 | 富马酸伏诺拉生| 1260141-27-2
英文名称 Vonoprazan Fumarate | TAK-438
CAS号881681-01-2
分子式C17H16FN3O2S· C4H4O4
分子量461.46 | 345.39 (Free)
外观White to off-white powder
储存条件4°C, sealed storage, away from moisture and light
安全信息
产品详情

Vonoprazan Fumarate, also known as TAK438, is a new medicine for treating acid-related diseases with a novel mechanism of action called potassium-competitive acid blockers (P-CABs) which competitively inhibits the binding of potassium ions to H+,K+-ATPase (also known as the proton pump) in the final step of gastric acid secretion in gastric parietal cells. TAKECAB provides a strong and sustained acid secretion inhibitory effect.

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