| 中文名称 | 氢溴酸卤夫酮 | 氢溴酸常山酮 | 氢溴酸溴氯哌喹酮 | 卤夫酮氢溴酸盐 | 常山酮氢溴酸盐 |
|---|---|
| 英文名称 | Halofuginone hydrobromide (Synonyms: RU-19110 hydrobromide) |
| CAS号 | 64924-67-0 |
| 分子式 | C16H18Br2ClN3O3 |
| 分子量 | 495.59 |
Halofuginone (RU-19110) hydrobromide, a Febrifugine derivative, is a competitive prolyl-tRNA synthetase inhibitor with a Ki of 18.3 nM. Halofuginone hydrobromid is a specific inhibitor of type-I collagen synthesis and attenuates osteoarthritis (OA) by inhibition of TGF-β activity. Halofuginone hydrobromid is also a potent pulmonary vasodilator by activating Kv channels and blocking voltage-gated, receptor-operated and store-operated Ca2+ channels. Halofuginone hydrobromid has anti-malaria, anti-inflammatory, anti-cancer, anti-fibrosis effects.
Tags: buy Halofuginone hydrobromide | Halofuginone hydrobromide supplier | purchase Halofuginone hydrobromide | Halofuginone hydrobromide cost | Halofuginone hydrobromide manufacturer | order Halofuginone hydrobromide | Halofuginone hydrobromide distributor
© 2020-2024 凯立德生物医药技术(上海)有限公司 版权所有
沪ICP备15046197号-3
沪公网安备31011502007856号
Designed by Kuanersoft