SB 271046 HCl | SB 271046A
SB 271046 Hydrochloride (Synonyms: SB 271046A)
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基本信息
中文名称SB 271046 HCl | SB 271046A
英文名称 SB 271046 Hydrochloride (Synonyms: SB 271046A)
CAS号209481-24-3
分子式C20H23Cl2N3O3S2
分子量488.45
储存条件4°C, sealed storage, away from moisture
安全信息
产品详情

SB 271046 Hydrochloride (SB 271046A) is a potent, selective and orally active 5-HT6 receptor antagonist with pKi of 9.02, 8.55, and 8.81 for rat, pig and human, respectively. SB 271046 Hydrochloride is over 200 fold selective for the 5-HT6 receptor vs 55 other receptors, binding sites and ion channels. Anticonvulsant activity (EC50=0.16 μM).
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