Olcegepant hydrochloride (BIBN-4096 hydrochloride; BIBN4096BS hydrochloride)
Olcegepant hydrochloride (Synonyms: BIBN-4096 hydrochloride; BIBN4096BS hydrochloride)
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基本信息
中文名称Olcegepant hydrochloride (BIBN-4096 hydrochloride; BIBN4096BS hydrochloride)
英文名称 Olcegepant hydrochloride (Synonyms: BIBN-4096 hydrochloride; BIBN4096BS hydrochloride)
CAS号586368-06-1
分子式C38H47Br2N9O5.HCl
分子量906.11
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Olcegepant hydrochloride (BIBN-4096 hydrochloride) is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and with a Ki of 14.4 pM for human CGRP.

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Olcegepant hydrochloride (BIBN-4096 hydrochloride; BIBN4096BS hydrochloride)