SNX 2112 | PF-04928473
SNX-2112 (Synonyms: PF-04928473)
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产品库存
3-5days
目录价格
¥668.00
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产品库存
3-5days
目录价格
¥998.00
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3-5days
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¥2860.00
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基本信息
中文名称SNX 2112 | PF-04928473
英文名称 SNX-2112 (Synonyms: PF-04928473)
CAS号908112-43-6
分子式C23H27F3N4O3
分子量464.48
外观White to off-white powder
储存条件Store in a dry and dark sealed container, short-term (weeks to months) storage at 0-4 ℃, long-term (months to years) storage at -20 ℃.
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产品详情

 SNX-2112, also known as PF 04928473, is an Hsp90 inhibitor which is currently undergoing multiple phase 1 clinical trials. In all cell lines, SNX-2112 led to degradation of MET, HER-2, EGFR, and AKT as well as abrogation of Ras/Raf/MEK/MAPK and PI3K/AKT signaling, followed by complete cell cycle arrest.

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