中文名称 | SB408124 HCl |
---|---|
英文名称 | SB-408124 Hydrochloride |
CAS号 | 1431697-90-3 |
分子式 | C19H18F2N4O·HCl |
分子量 | 392.83 | 356.38(free) |
外观 | White to gray powder |
储存条件 | 4°C, sealed storage, away from moisture |
SB-408124 Hydrochloride is a selective non-peptide orexin receptor 1 (OX1) receptor antagonist with Kis of 57 nM and 27 nM in whole cell and membrane, respectively. SB-408124 Hydrochloride exhibits 50-fold selectivity over OX2 receptor.
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