中文名称 | 他克莫司 |
---|---|
英文名称 | Tacrolimus | Fujimycin | FR900506 | FK506 |
CAS号 | 104987-11-3 |
分子式 | C44H69NO12 |
分子量 | 804.02 |
外观 | White to off-white powder |
储存条件 | 4°C, protect from light |
Tacrolimus (FK506), a macrocyclic lactone, binds to FK506 binding protein (FKBP) to form a complex. Tacrolimus inhibits calcineurin phosphatase, which inhibits T-lymphocyte signal transduction and IL-2 transcription. Immunosuppressive properties.
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