| 中文名称 | N1-羟基-N8-苯基辛二酰胺; 伏立诺他 | 伏瑞斯特 |
|---|---|
| 英文名称 | Vorinostat (SAHA) (Synonyms: MK0683; Suberoylanilide hydroxamic acid) |
| CAS号 | 149647-78-9 |
| 分子式 | C14H20N2O3 |
| 分子量 | 264.3 |
| MDL | MFCD00945317 |
| 外观 | White or off-white powder |
| 储存条件 | Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years). |
Vorinostat (SAHA) is an HDAC inhibitor with IC50 of ~10 nM in a cell-free assay. Vorinostat abrogates productive HPV-18 DNA amplification.
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