帕潘立酮棕榈酸酯
Paliperidone Palmitate (Synonyms: 9-Hydroxyrisperidone Palmitate)
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基本信息
中文名称帕潘立酮棕榈酸酯
英文名称 Paliperidone Palmitate (Synonyms: 9-Hydroxyrisperidone Palmitate)
CAS号199739-10-1
分子式C39H57FN4O4
分子量664.89
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Paliperidone palmitate is an orally effective competitive antagonist of dopamine D2 receptors and 5-hydroxytryptamine 2A (5-HT2A) receptors that can cross the blood-brain barrier. Paliperidone palmitate competitively inhibits the effects of dopamine and 5-hydroxytryptamine by binding to dopamine D2 receptors and 5-HT2A receptors, regulating the balance of the neurotransmitter system and thus exerting antipsychotic activity. Paliperidone palmitate is mainly used in the research field of schizophrenia.
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