中文名称 | (S)-3-(((3-乙基-5-(2-(2-羟乙基)哌啶-1-基)吡唑并[1,5-a]嘧啶-7-基)氨基)甲基)吡啶 1-氧化物 |
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英文名称 | Dinaciclib (Synonyms: SCH 727965; SCH727965; PS-095760) |
CAS号 | 779353-01-4 |
分子式 | C21H28N6O2 |
分子量 | 396.49 |
Dinaciclib (SCH 727965) is a potent inhibitor of CDK, with IC50s of 1 nM, 1 nM, 3 nM, and 4 nM for CDK2, CDK5, CDK1, and CDK9, respectively.
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