乌帕替尼半水合物
Upadacitinib hemihydrate
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中文名称乌帕替尼半水合物
英文名称 Upadacitinib hemihydrate
CAS号2050057-56-0
分子式C34H40F6N12O3
分子量778.75
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Upadacitinib, also known as ABT-494, is a potent and selective JAK inhibitors in development for rheumatoid arthritis. ABT-494 is approximately 74 fold selective for Jak1 over Jak2 in cellular assays dependent on specific, relevant cytokines. ABT-494 demonstrates efficacy in rat arthritis models. Preliminary evidence suggests that compared to tofacitinib, ABT-494 may spare Jak2 and Jak3 dependent signaling.

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乌帕替尼半水合物