中文名称 | 甲磺酸乐伐替尼 | 仑伐替尼甲酸盐 |
---|---|
英文名称 | Lenvatinib Mesylate | E7080 mesylate | ER-203492-00 |
CAS号 | 857890-39-2 |
分子式 | C21H19ClN4O4.CH4O3S |
分子量 | 522.96 |
外观 | Off-white powder |
储存条件 | Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years). |
Lenvatinib Mesylate is a synthetic, orally available tyrosine kinase inhibitor that inhibits vascular endothelial growth factor receptor (VEGFR1-3), fibroblast growth factor receptor (FGFR1-4), platelet-derived growth factor receptor α (PDGFRα), stem cell factor receptor (Kit (c-Kit)), and rearranged during transfection (RET (c-RET)). Lenvatinib Mesylate has potential antineoplastic activity.
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