甲磺酸乐伐替尼 | 仑伐替尼甲酸盐
Lenvatinib Mesylate (Synonyms: E7080 mesylate; ER-203492-00)
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基本信息
中文名称甲磺酸乐伐替尼 | 仑伐替尼甲酸盐
英文名称 Lenvatinib Mesylate (Synonyms: E7080 mesylate; ER-203492-00)
CAS号857890-39-2
分子式C21H19ClN4O4.CH4O3S
分子量522.96
外观Off-white powder
储存条件Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years).
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Lenvatinib Mesylate is a synthetic, orally available tyrosine kinase inhibitor that inhibits vascular endothelial growth factor receptor (VEGFR1-3), fibroblast growth factor receptor (FGFR1-4), platelet-derived growth factor receptor α (PDGFRα), stem cell factor receptor (Kit (c-Kit)), and rearranged during transfection (RET (c-RET)). Lenvatinib Mesylate has potential antineoplastic activity.
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