中文名称 | SX 011/SX-011 |
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英文名称 | SX 011/SX-011 |
CAS号 | 309913-42-6 |
分子式 | C26H27ClFN3O3 |
分子量 | 483.96 |
外观 | White to off-white powder |
储存条件 | Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years). |
SX-011 is a p38 inhibitor with IC50 values for p38 and p38β of 9 nM and 90 nM, respectively. Additionally, SX-011 blocks JNK-2 with an IC50 of 100 nM. Orally, SX-011 is bioavailable.
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