中文名称 | 格佐匹韦 | 格拉瑞韦 |
---|---|
英文名称 | Grazoprevir (Synonyms: MK-5172) |
CAS号 | 1350514-68-9 |
分子式 | C38H50N6O9S |
分子量 | 766.90 |
Grazoprevir (MK-5172) is a selective inhibitor of Hepatitis C virus NS3/4a protease with broad activity across genotypes and resistant variants, with Kis of 0.01 nM (gt1b), 0.01 nM (gt1a), 0.08 nM (gt2a), 0.15 nM (gt2b), 0.90 nM (gt3a), respectively. Grazoprevir inhibits SARS-CoV-2 3CLpro activity.
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