赛乐西帕 | 司来帕格
Selexipag (Synonyms: NS-304; ACT-293987)
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3-5days
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¥300.00
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3-5days
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¥500.00
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3-5days
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¥800.00
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基本信息
中文名称赛乐西帕 | 司来帕格
英文名称 Selexipag (Synonyms: NS-304; ACT-293987)
CAS号475086-01-2
分子式C26H32N4O4S
分子量496.62
外观 White to yellow powder
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Selexipag, also known as ACT-293987 and NS-304, is a a first-in-class orally available selective non-prostanoid IP receptor agonist, which is currently in development by Actelion as a treatment of pulmonary arterial hypertension. Selexipag and its active metabolite, ACT-333679, are agonists at the prostacyclin receptor, which leads to vasodilation in the pulmonary circulation.

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