奥西卓司他
Osilodrostat (Synonyms: LCI699)
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产品库存
3-5days
目录价格
¥350.00
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产品库存
3-5days
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¥660.00
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3-5days
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¥1150.00
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基本信息
中文名称奥西卓司他
英文名称 Osilodrostat (Synonyms: LCI699)
CAS号928134-65-0
分子式C13H10FN3
分子量227.24
外观White to yellow pwder
储存条件Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years).
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Osilodrostat, also known as LCI699, is a potent inhibitor of 11β-hydroxylase, the enzyme which catalyzes the final step of cortisol synthesis. LCI699 may thus be a potential new treatment for all forms of Cushing's syndrome. Current evidence indicates that the novel aldosterone inhibitor LCI699 is an effective and well-tolerated antihypertensive agent that lowers plasma aldosterone concentration and produces a mild ACTH-stimulated cortisol response suppressive effect.
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Osilodrostat phosphate(LCI699 phosphate)
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