玛伐凯泰 | 马瓦卡坦
Mavacamten (Synonyms: MYK461; SAR439152;MYK-461)
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基本信息
中文名称玛伐凯泰 | 马瓦卡坦
英文名称 Mavacamten (Synonyms: MYK461; SAR439152;MYK-461)
CAS号1642288-47-8
分子式C15H19N3O2
分子量273.33
外观White to off-white powder
储存条件Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years).
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 Mavacamten, also known as SAR-439152 and MYK-461, is a myosin inhibitor potentially for the treatment of hypertrophic cardiomyopathy. SAR-439152 reduces contractility by decreasing the adenosine triphosphatase activity of the cardiac myosin heavy chain.
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