中文名称 | 盐酸罗匹尼罗 |
---|---|
英文名称 | Ropinirole hydrochloride (Synonyms: Ropinirole HCl; SKF 101468 hydrochloride;SKF-101468A) |
CAS号 | 91374-20-8 |
分子式 | C16H25ClN2O |
分子量 | 296.84 |
外观 | White to yellow powder |
储存条件 | 4°C, sealed storage, away from moisture |
Ropinirole (SKF 101468) hydrochloride is an orally active, potent D3/D2 receptor agonist with a Ki of 29 nM for D2 receptor. Ropinirole hydrochloride has pEC50s of 7.4, 8.4 and 6.8 for hD2, hD3 and hD4 receptors, respectively. Ropinirole hydrochloride has no affinity for the D1 receptors. Ropinirole hydrochloride has the potential for Parkinson's disease.
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