| 中文名称 | N-(5-(4-氰基苯基)-1H-吡咯并[2,3-b]吡啶-3-基)吡啶-3-甲酰胺 |
|---|---|
| 英文名称 | Pim1/AKK1-IN-1 (Synonyms: LKB1/AAK1 dual inhibitor) |
| CAS号 | 1093222-27-5 |
| 分子式 | C20H13N5O |
| 分子量 | 339.35 |
| MDL | MFCD15528944 |
| 外观 | White to gray powder |
| 储存条件 | Store short-term at 0-4°C or long-term at -20°C in a dry, dark place. |
Pim1/AKK1-IN-1 is a potent multi-kinase inhibitor with Kd values of 35 nM/53 nM/75 nM/380 nM for Pim1/AKK1/MST2/LKB1 respectively, and it also inhibits MPSK1 and TNIK.
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