中文名称 | N-(5-(4-氰基苯基)-1H-吡咯并[2,3-b]吡啶-3-基)吡啶-3-甲酰胺 |
---|---|
英文名称 | Pim1/AKK1-IN-1 (Synonyms: LKB1/AAK1 dual inhibitor) |
CAS号 | 1093222-27-5 |
分子式 | C20H13N5O |
分子量 | 339.35 |
MDL | MFCD15528944 |
外观 | White to gray powder |
储存条件 | Store short-term at 0-4°C or long-term at -20°C in a dry, dark place. |
Pim1/AKK1-IN-1 is a potent multi-kinase inhibitor with Kd values of 35 nM/53 nM/75 nM/380 nM for Pim1/AKK1/MST2/LKB1 respectively, and it also inhibits MPSK1 and TNIK.
© 2020-2024 凯立德生物医药技术(上海)有限公司 版权所有
沪ICP备15046197号-3
沪公网安备31011502007856号
Designed by Kuanersoft