Obicetrapib (TA-8995; DEZ-001)
Obicetrapib (Synonyms: TA-8995; DEZ-001)
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产品库存
3-5 days
目录价格
¥1288.00
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产品库存
3-5 days
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¥1936.00
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产品库存
3-5 days
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¥2996.00
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产品库存
3-5 days
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¥4788.00
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基本信息
中文名称Obicetrapib (TA-8995; DEZ-001)
英文名称 Obicetrapib (Synonyms: TA-8995; DEZ-001)
CAS号866399-87-3
分子式C32H31F9N4O5
分子量722.60
MDL MFCD30533470
外观White to light yellow powder
储存条件Store short-term at 0-4°C or long-term at -20°C in a dry, dark place.
安全信息
产品详情

Obicetrapib, also known as AMG-899, TA-8995, and DEX-001, is a cholesteryl ester transfer protein (CETP) inhibitor. CETP inhibitors substantially increase the concentration of high-density lipoprotein cholesterol (HDL-C), which may have a possible beneficial effect for cardiovascular disease risk reduction. TA-8995 dose dependently increased not only total and non-ABCA1-specific CEC but also ABCA1-specific CEC and preBeta-1 HDL particle levels.

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