中文名称 | 6-(3-氨基苄基)-4-甲基-2-(甲基亚磺酰基)-4H-噻吩并[2',3':4,5]吡咯并[2,3-d]哒嗪-5(6H)-酮 |
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英文名称 | TEPP-46 (Synonyms: ML-265) |
CAS号 | 1221186-53-3 |
分子式 | C17H16N4O2S2 |
分子量 | 372.46 |
MDL | MFCD23160747 |
外观 | White to light yellow powder |
储存条件 | Store short-term at 0-4°C or long-term at -20°C in a dry, dark place. |
TEPP-46, also known as ML265, is a potent and selective PKM2 activator with an AC50 of 92 nM, exhibiting high selectivity over PKM1, PKR, and PKL.
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