SB-742457 (GSK-742457; RVT-101; Intepirdine)
Intepirdine (Synonyms: SB-742457; GSK-742457; RVT-101)
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基本信息
中文名称SB-742457 (GSK-742457; RVT-101; Intepirdine)
英文名称 Intepirdine (Synonyms: SB-742457; GSK-742457; RVT-101)
CAS号607742-69-8
分子式C19H19N3O2S
分子量353.44
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Intepirdine (SB742457) is a highly selective 5-HT6 receptor antagonist with pKi of 9.63; exhibits >100-fold selectivity over other receptors.
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SB-742457 (GSK-742457; RVT-101; Intepirdine)