依洛尤单抗; 依伏库单抗
Anti-Human PCSK9 Monoclonal Antibody(Evolocumab); AMG 145
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1 mg 5 mg 10 mg 50 mg 100 mg
产品库存
3-5days
目录价格
¥3000.00
会员价格
产品库存
3-5days
目录价格
¥12500.00
会员价格
产品库存
3-5days
目录价格
¥20000.00
会员价格
产品库存
3-5days
目录价格
¥80000.00
会员价格
产品库存
3-5days
目录价格
¥125000.00
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- +
基本信息
中文名称依洛尤单抗; 依伏库单抗
英文名称 Anti-Human PCSK9 Monoclonal Antibody(Evolocumab); AMG 145
CAS号1256937-27-5
外观Colorless to light yellow (Solution)
储存条件Store the undiluted solution at 4°C in the dark to avoid freeze-thaw cycles.
安全信息
产品详情

Evolocumab (AMG 145) is a human monoclonal antibody that inhibits PCSK9. Evolocumab is used in the study of hypercholesterolemia and atherosclerotic cardiovascular disease. Evolocumab binds to circulating PCSK9 protein and inhibits its binding to LDLR. Evolocumab has antioxidant and cytoprotective activities against H2O2-induced oxidative damage to endothelial cells. Evolocumab may also negatively regulate activation of the TLR-4/NF-κB signaling pathway to prevent inflammation.

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依洛尤单抗; 依伏库单抗