GSK2606414;GSK 2606414

规格	库存	目录价	会员专享价	数量
20 mg	3-5days	￥520.00	登录后可见	- +
50 mg	3-5days	￥850.00	登录后可见	- +
100 mg	3-5days	￥1450.00	登录后可见	- +

规格

库存

目录价

会员专享价

数量

20 mg

3-5days

￥520.00

登录后可见

- +

50 mg

3-5days

￥850.00

登录后可见

- +

100 mg

3-5days

￥1450.00

登录后可见

- +

基本信息

英文名称	GSK2606414;GSK 2606414
中文名称	GSK2606414;GSK 2606414
CAS号	1337531-36-8
分子式	C24H20F3N5O
分子量	451.44
外观	white powder
储存条件	Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years).

产品详情

GSK2606414 is an orally available, selective protein kinase R-like ER kinase (PERK) inhibitor with an IC₅₀ value of 0.4 nM. It can inhibit thapsigargin-induced PERK phosphorylation in lung carcinoma A549 cells and attenuates subcutaneous pancreatic human tumor xenograft growth in mice. Because PERK mediates the unfolded protein response pathway, which has roles in neurotoxicity and cancer, inhibition of PERK signaling has potential applications for the treatment of cancer and also cognitive degeneration.

GSK2606414;GSK 2606414

GSK2606414;GSK 2606414

化学品安全说明书(MSDS)

质检证书(COA)