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Catalog No：CL2099 CAS No.：168273-06-1 MDLNo： Formula：C22H21Cl3N4O MW：463.79

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Size	Availability	Price(USD)	VIP Price (USD)	Quantity
25 mg	3-5days	￥206.00	Visible after login	- +
50 mg	3-5days	￥348.00	Visible after login	- +

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Product Overview

Product Name	Rimonabant \| SR141716
CAS	168273-06-1
Formula	C22H21Cl3N4O
MW	463.79
Appearance	White to off-white powder
Storage condition	4°C, sealed storage, away from moisture

Product details

Rimonabant (SR141716) is a highly potent, brain penetrated and selective central cannabinoid receptor (CB1) antagonist with a K_i of 1.8 nM. Rimonabant (SR141716) also inhibits Mycobacterial membrane protein Large 3 (MMPL3).

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AM-251 and rimonabant act as direct antagonists at mu-opioid receptors: Implications for opioid/cannabinoid interaction studies.

PMID: 22771770 PMCID: PMC3408547 DOI: 10.1016/j.neuropharm.2012.06.046

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The inverse agonist effect of rimonabant on G protein activation is not mediated by the cannabinoid CB1 receptor: Evidence from postmortem human brain.

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