Linsitinib (OSI-906)

Size	Availability	Price(USD)	VIP Price (USD)	Quantity
1 mg	3-5days	￥500.00	Visible after login	- +
5 mg	3-5days	￥980.00	Visible after login	- +
10 mg	3-5days	￥1600.00	Visible after login	- +

Size

Availability

Price(USD)

VIP Price (USD)

Quantity

1 mg

3-5days

￥500.00

Visible after login

- +

5 mg

3-5days

￥980.00

Visible after login

- +

10 mg

3-5days

￥1600.00

Visible after login

- +

Product Overview

Product Name	Linsitinib (OSI-906)
CAS	867160-71-2
Formula	C26H23N5O
MW	421.49
Appearance	White to yellow powder
Storage condition	Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years).

Product details

Linsitinib (formerly OSI-906; OSI 906) is a firs-in-class, ATP-competitive and orally bioavailable dual inhibitor of and insulin receptor (IR) and insulin-like growth factor-1 receptor (IGF-1R) with potential antitumor activity. It exhibits modest potency against InsR with an IC50 of 75 nM, and it has no activity against other kinases like Abl, ALK, BTK, EGFR, FGFR1/2, PKA, and so on. In cell-free assays, it inhibits IGF-1R with an IC50 of 35 nM.

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