PD 168368

Size	Availability	Price(USD)	VIP Price (USD)	Quantity
1 mg	3-5days	￥968.00	Visible after login	- +
5 mg	3-5days	￥3866.00	Visible after login	- +

Size

Availability

Price(USD)

VIP Price (USD)

Quantity

1 mg

3-5days

￥968.00

Visible after login

- +

5 mg

3-5days

￥3866.00

Visible after login

- +

Product Overview

Product Name	PD 168368
CAS	204066-82-0
Formula	C31H34N6O4
MW	554.64
Appearance	White to off-white powder
Storage condition	Store in a dry and dark sealed container, short-term (weeks to months) storage at 0-4 ℃, long-term (months to years) storage at -20 ℃.

Product details

PD 168368 is a novel, potent, competitive and selective nonpeptide neuromodulin B receptor (NMB-R) antagonist with inhibitory effects on the gastrin-releasing peptide receptor (GRPR).PD 168368 is a potent mixed agonist of FPR1/FPR2/FPR3.

Related literature

Tyrosine 220 in the 5th transmembrane domain of the neuromedin B receptor is critical for the high selectivity of the peptoid antagonist PD168368.

PMID: 11013243 DOI: 10.1074/jbc.M006059200

Comparative pharmacology of the nonpeptide neuromedin B receptor antagonist PD 168368.

PMID: 10454496

Gastrin-releasing peptide/neuromedin B receptor antagonists PD176252, PD168368, and related analogs are potent agonists of human formyl-peptide receptors.

PMID: 20943772 PMCID: PMC3014281 DOI: 10.1124/mol.110.068288

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