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(2E)-N-[4-[3-氯-4-(2-吡啶基甲氧基)苯胺基]-3-氰基-7-乙氧基-6-喹啉基]-4-(二甲氨基)-2-丁烯酰胺；来那替尼

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Catalog No：CL2190 CAS No.：698387-09-6 MDLNo：MFCD09752958 Formula：C30H29ClN6O3 MW：557.04

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Size	Availability	Price(USD)	VIP Price (USD)	Quantity
100 mg	In-stock	￥426.00	Visible after login	- +
200 mg	In-stock	￥736.00	Visible after login	- +
500 mg	In-stock	￥1386.00	Visible after login	- +

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Product Overview

Product Name	Neratinib (Synonyms: HKI-272)
CAS	698387-09-6
Formula	C30H29ClN6O3
MW	557.04
MDL	MFCD09752958
Appearance	Pale yellow to white powder
Storage condition	Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years).

Product details

Neratinib is a highly selective inhibitor of HER2 and EGFR, demonstrating IC50 values of 59 nM and 92 nM in cell-free assays, respectively. It weakly inhibits KDR and Src, while showing no significant inhibition against Akt, CDK1/2/4, IKK-2, MK-2, PDK1, c-Raf, and c-Met.

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CL2190

Neratinib (Synonyms: HKI-272)

698387-09-6 98+%