Preladenant | SCH 420814 | 377727-87-2

Size	Availability	Price(USD)	VIP Price (USD)	Quantity
10 mg	In-stock	￥366.00	Visible after login	- +
25 mg	In-stock	￥656.00	Visible after login	- +
50 mg	3-5days	￥1068.00	Visible after login	- +

Size

Availability

Price(USD)

VIP Price (USD)

Quantity

10 mg

In-stock

￥366.00

Visible after login

- +

25 mg

In-stock

￥656.00

Visible after login

- +

50 mg

3-5days

￥1068.00

Visible after login

- +

Product Overview

Product Name	Preladenant \| SCH 420814
CAS	377727-87-2
Formula	C25H29N9O3
MW	503.56
Appearance	White to off-white powder
Storage condition	Store in a dry and dark sealed container, short-term (weeks to months) storage at 0-4 ℃, long-term (months to years) storage at -20 ℃.

Product details

Preladenant is a potent and competitive antagonist of the human adenosine A2A receptor with a K_i of 1.1 nM and has over 1000-fold selectivity over other adenosine receptors.

Related literature

Characterization of the potent and highly selective A2A receptor antagonists preladenant and SCH 412348 [7-[2-[4-2,4-difluorophenyl]-1-piperazinyl]ethyl]-2-(2-furanyl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine] in rodent models of movement disorders and depression.

PMID: 19332567 DOI: 10.1124/jpet.108.149617

Preladenant, a selective A(2A) receptor antagonist, is active in primate models of movement disorders.

PMID: 20655910 DOI: 10.1016/j.expneurol.2010.07.011

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History

CL2394

Preladenant | SCH 420814

377727-87-2 98+%

CL2869A

Streptomycin | Agrept | Agrimycin | Streptomycin A

57-92-1 98+%

瑞德南特

Chemical safety data sheet(MSDS)

Certificate Of Authenticity(CPA)