Dovitinib lactate hydrate (Synonyms: TKI258 lactate hydrate; CHIR-258 lactate hydrate) ; CAS: 915769-50-5

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Product Overview

Product Name	Dovitinib (TKI258) Lactate monohydrate (Synonyms: TKI258 lactate hydrate; CHIR-258 lactate hydrate;CHIR258)
CAS	915769-50-5
Formula	C24H29FN6O5
MW	500.52
MDL	MFCD16038433
Appearance	Light yellow to yellow powder
Storage condition	4°C, sealed storage, away from moisture

Product details

Dovitinib lactate hydrate (TKI258 lactate hydrate) is a potent multi-targeted tyrosine kinase inhibitor with IC50 values of 1 nM for FLT3, 2 nM for c-Kit, 8-9 nM for FGFR1/3, 10-13 nM for VEGFR1/2/3, and 27-210 nM for PDGFRα/β, respectively.

Related literature

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