Home > Category > Signaling Pathways > JAK/STAT Signaling > Pim > Pim1/AKK1-IN-1 (Synonyms: LKB1/AAK1 dual inhibitor)

N-(5-(4-氰基苯基)-1H-吡咯并[2,3-b]吡啶-3-基)吡啶-3-甲酰胺

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Catalog No：CL3110 CAS No.：1093222-27-5 MDLNo：MFCD15528944 Formula：C20H13N5O MW：339.35

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Product Overview

Product Name	Pim1/AKK1-IN-1 (Synonyms: LKB1/AAK1 dual inhibitor)
CAS	1093222-27-5
Formula	C20H13N5O
MW	339.35
MDL	MFCD15528944
Appearance	White to gray powder
Storage condition	Store short-term at 0-4°C or long-term at -20°C in a dry, dark place.

Product details

Pim1/AKK1-IN-1 is a potent multi-kinase inhibitor with Kd values of 35 nM/53 nM/75 nM/380 nM for Pim1/AKK1/MST2/LKB1 respectively, and it also inhibits MPSK1 and TNIK.

Related literature

Assessment of chemical coverage of kinome space and its implications for kinase drug discovery.

PMID: 19035792 DOI: 10.1021/jm8011036

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CL3110

Pim1/AKK1-IN-1 (Synonyms: LKB1/AAK1 dual inhibitor)

1093222-27-5 98+%