| 英文名称 | Cobimetinib Hemifumarate (Synonyms: GDC-0973 hemifumarate; XL-518 hemifumarate) |
|---|---|
| 中文名称 | 考比替尼半富马酸盐 |
| CAS号 | 1369665-02-0 |
| 分子式 | C21H21F3IN3O2·1/2C4H4O4 |
| 分子量 | 589.25 |
| MDL | MFCD31544353 |
| 外观 | White to off-white powder |
| 储存条件 | 4°C, sealed storage, away from moisture |
| 英文名称 | Cobimetinib Hemifumarate (Synonyms: GDC-0973 hemifumarate; XL-518 hemifumarate) |
|---|---|
| 中文名称 | 考比替尼半富马酸盐 |
| CAS号 | 1369665-02-0 |
| 分子式 | C21H21F3IN3O2·1/2C4H4O4 |
| 分子量 | 589.25 |
| MDL | MFCD31544353 |
| 外观 | White to off-white powder |
| 储存条件 | 4°C, sealed storage, away from moisture |
Cobimetinib hemifumarate is a novel selective MEK1 inhibitor, and the IC50 value against MEK1 is 4.2 nM.
Tags: buy Cobimetinib Hemifumarate (GDC-0973 hemifumarate) | Cobimetinib Hemifumarate (GDC-0973 hemifumarate) supplier | purchase Cobimetinib Hemifumarate (GDC-0973 hemifumarate) | Cobimetinib Hemifumarate (GDC-0973 hemifumarate) cost | Cobimetinib Hemifumarate (GDC-0973 hemifumarate) manufacturer | orderCobimetinib Hemifumarate (GDC-0973 hemifumarate) | Cobimetinib Hemifumarate (GDC-0973 hemifumarate) distributor
PMID: 23053270 DOI: 10.1007/s00280-012-1988-6
PMID: 22084396 DOI: 10.1158/0008-5472.CAN-11-1515
PMID: 22496205 DOI: 10.1158/1078-0432.CCR-12-0445
PMID: 27250023 PMCID: PMC5129946 DOI: 10.18632/oncotarget.7790