英文名称 | PND-1186 hydrochloride (Synonyms: VS-4718 hydrochloride; SR-2516 hydrochloride) |
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中文名称 | PND-1186 hydrochloride |
CAS号 | 1356154-94-3 |
分子式 | C25H27ClF3N5O3 |
分子量 | 537.96 |
英文名称 | PND-1186 hydrochloride (Synonyms: VS-4718 hydrochloride; SR-2516 hydrochloride) |
---|---|
中文名称 | PND-1186 hydrochloride |
CAS号 | 1356154-94-3 |
分子式 | C25H27ClF3N5O3 |
分子量 | 537.96 |
PND-1186 hydrochloride (VS-4718 hydrochloride) is a potent, highly-specific and reversible inhibitor of FAK with an IC50 of 1.5 nM. PND-1186 hydrochloride selectively promotes tumor cell apoptosis.