Pelabresib | CPI-0610 | 1380087-89-7

规格	库存	目录价	会员专享价	数量
5 mg	In-stock	￥1100.00	登录后可见	- +
10 mg	In-stock	￥2100.00	登录后可见	- +

规格

库存

目录价

会员专享价

数量

5 mg

In-stock

￥1100.00

登录后可见

- +

10 mg

In-stock

￥2100.00

登录后可见

- +

基本信息

英文名称	Pelabresib (Synonyms: CPI-0610)
中文名称	(S)-2-(6-(4-氯苯基)-1-甲基-4H-苯并[c]异恶唑并[4,5-e]氮杂环庚烷-4-基)乙酰胺
CAS号	1380087-89-7
分子式	C20H16ClN3O2
分子量	365.81
MDL	MFCD28144505
外观	White to off-white powder
储存条件	Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years).

产品详情

Pelabresib (CPI-0610) is a potent and selective benzoisoxazoloazepine BET bromodomain inhibitor with an IC50 of 39 nM for BRD4-BD1 in TR-FRET assay and currently undergoing human clinical trials for hematological malignancies. CPI-0610 inhibits the expression of Nuclear receptor binding SET domain protein 3 (NSD3) target genes.

(S)-2-(6-(4-氯苯基)-1-甲基-4H-苯并[c]异恶唑并[4,5-e]氮杂环庚烷-4-基)乙酰胺

Pelabresib (Synonyms: CPI-0610)

化学品安全说明书(MSDS)

质检证书(COA)