| 英文名称 | Tariquidar methanesulfonate, hydrate | XR9576 methanesulfonate, hydrate |
|---|---|
| 中文名称 | 他立喹达二甲磺酸盐水合物 |
| CAS号 | 625375-83-9 |
| 分子式 | C38H38N4O6 · 2CH4O3S · 3H2O |
| 分子量 | 892.99 | 646.74 (free) |
| 外观 | Light yellow to yellow powder |
| 储存条件 | 4°C, sealed storage, away from moisture |
| 英文名称 | Tariquidar methanesulfonate, hydrate | XR9576 methanesulfonate, hydrate |
|---|---|
| 中文名称 | 他立喹达二甲磺酸盐水合物 |
| CAS号 | 625375-83-9 |
| 分子式 | C38H38N4O6 · 2CH4O3S · 3H2O |
| 分子量 | 892.99 | 646.74 (free) |
| 外观 | Light yellow to yellow powder |
| 储存条件 | 4°C, sealed storage, away from moisture |
Tariquidar methanesulfonate, hydrate (XR9576 methanesulfonate, hydrate) is a potent and specific inhibitor of P-glycoprotein (P-gp) with a Kd of 5.1 nM.