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替氟朵

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Catalog No:CL1856 CAS No.:83386-35-0 MDLNo: Formula:C22H20FN3OS MW:393.48
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Product Overview
Product Name Tifluadom | KC 5103 | dl-Tifluadom
CAS83386-35-0
FormulaC22H20FN3OS
MW393.48
Storage conditionStore in a dry and dark sealed container, short-term (weeks to months) storage at 0-4 ℃, long-term (months to years) storage at -20 ℃.
Product details

Tifluadom is a kappa-opioid receptor agonist. It has been shown to produce antinociception in the rotarod test and locomotor activity in mice, as well as having other pharmacological effects. Tifluadom is used to treat inflammatory disorders and autoimmune diseases. The mechanism of action of Tifluadom is not fully understood, but it may be due to its ability to bind with the benzodiazepine binding site on the GABAA receptor and also activate κ-opioid receptors. Tifluadom has been shown to increase the glomerular filtration rate (GFR) in rats by activating dopaminergic receptors that are involved in renal function.


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