| 英文名称 | Brivanib Alaninate (Synonyms: BMS-582664) |
|---|---|
| 中文名称 | 丙氨酸布立尼布 |
| CAS号 | 649735-63-7 |
| 分子式 | C22H24FN5O4 |
| 分子量 | 441.46 |
| 英文名称 | Brivanib Alaninate (Synonyms: BMS-582664) |
|---|---|
| 中文名称 | 丙氨酸布立尼布 |
| CAS号 | 649735-63-7 |
| 分子式 | C22H24FN5O4 |
| 分子量 | 441.46 |
Brivanib alaninate (BMS-582664) is an ATP-competitive inhibitor against VEGFR2 with an IC50 of 25 nM; has moderate potency against VEGFR-1 and FGFR-1, but more than 240-fold against PDGFRβ.
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PMID: 16570908 DOI: 10.1021/jm051106d
PMID: 26528545 PMCID: PMC4631495 DOI: 10.1371/journal.pone.0142355